Description：

AGI-5198 is the first highly potent and selective inhibitor of IDH1 R132H/R132C mutants with IC50 of 0.07 μM/0.16 μM.

Chemical Information：

Molecular Weight (MW)		462.56
Formula		C27H31FN4O2
CAS No.		1355326-35-0
Solubility (25°C) *	DMSO	24 mg/mL (51.88 mM)
	Water	Insoluble
	Alcohol	14 mg/mL (30.26 mM)

Biological Activity：

Targets IC50

ATM ATM 2.2 nM (Ki) 13 nM

Preparing Stock Solutions

Concentration Volume (DMSO) Mass	1 mg	5 mg	10 mg
1 mM	2.1619 mL	10.8094 mL	21.6188 mL
5 mM	0.4324 mL	2.1619 mL	4.3238 mL
10 mM	0.2162 mL	1.0809 mL	2.1619 mL
50 mM	0.0432 mL	0.2162 mL	0.4324 mL

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