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CGP 57380

CGP 57380

Catalog Number: CC7577 Rank: comment rank 5

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$ 130.00
$ 81.00
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Description:

CGP 57380 is a potent MNK1 inhibitor with IC50 of 2.2 μM, exhibiting no inhibitory activity on p38, JNK1, ERK1 and -2, PKC, or c-Src-like kinases.

Chemical Information:

Molecular Weight (MW) 244.23
Formula

 

C11H9FN6

 

CAS No. 522629-08-9
Solubility (25°C) * DMSO 48 mg/mL warmed (196.53 mM)
Water Insoluble
Alcohol Insoluble


Biological Activity:

Targets
IC50
p-Abl1T315I u-Abl1native u-Abl1T315I p-Abl1native Abl1H396P
4 nM 0.8 nM 5 nM 2 nM 1.4 nM


Preparing Stock Solutions

Concentration Volume (DMSO) Mass 1 mg 5 mg 10 mg
1 mM 4.0945 mL 20.4725 mL 40.9450 mL
5 mM 0.8189 mL 4.0945 mL 8.1890 mL
10 mM 0.4095 mL 2.0473 mL 4.0945 mL
50 mM 0.0819 mL 0.4095 mL 0.8189 mL


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