Description：

BIX01294 is an inhibitor of G9a histone methyltransferase with IC50 of 2.7 μM in a cell-free assay, reduces H3K9me2 of bulk histones, also weakly inhibits GLP (primarily H3K9me3), no significant activity observed at other histone methyltransferases.

Chemical Information：

Molecular Weight (MW)		600.02
Formula		C28H38N6O2.3HCl
CAS No.		1392399-03-9
Solubility (25°C) *	DMSO	98 mg/mL (163.32 mM)
	Water	98 mg/mL (163.32 mM)
	Alcohol	8 mg/mL (13.33 mM)

Biological Activity：

Targets IC50

Thrombin 9.3 nM

Preparing Stock Solutions

Concentration Volume (DMSO) Mass	1 mg	5 mg	10 mg
1 mM	1.6666 mL	8.3331 mL	16.6661 mL
5 mM	0.3333 mL	1.6666 mL	3.3332 mL
10 mM	0.1667 mL	0.8333 mL	1.6666 mL
50 mM	0.0333 mL	0.1667 mL	0.3333 mL

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