Description：

Tazemetostat (EPZ-6438) is a potent, and selective EZH2 inhibitor with K_i and IC50 of 2.5 nM and 11 nM in cell-free assays, exhibiting a 35-fold selectivity versus EZH1 and >4,500-fold selectivity relative to 14 other HMTs.

Chemical Information：

Molecular Weight (MW)		572.74
Formula		C34H44N4O4
CAS No.		1403254-99-8
Solubility (25°C) *	DMSO	5 mg/mL warmed (8.72 mM)
	Water	Insoluble
	Alcohol	Insoluble

Preparing Stock Solutions

Concentration Volume (DMSO) Mass	1 mg	5 mg	10 mg
1 mM	1.7460 mL	8.7300 mL	17.4599 mL
5 mM	0.3492 mL	1.7460 mL	3.4920 mL
10 mM	0.1746 mL	0.8730 mL	1.7460 mL
50 mM	0.0349 mL	0.1746 mL	0.3492 mL

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