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Anacetrapib (MK-0859)

Anacetrapib (MK-0859)

Catalog Number: CC2904 Rank: comment rank 5

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$ 189.00
$ 259.00
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Description:

Anacetrapib (MK0859) is a potent, selective, reversible rhCETP and mutant CETP(C13S) inhibitor with IC50 of 7.9 nM and 11.8 nM, increases HDL-C and decreases LDL-C, does not increase aldosterone or blood pressure. Phase 3.

Chemical Information:

Molecular Weight (MW) 637.51
Formula

 

C30H25F10NO3

 

CAS No. 875446-37-0
Solubility (25°C) * DMSO 127 mg/mL (199.21 mM)
Water Insoluble
Alcohol 127 mg/mL (199.21 mM)


Biological Activity:

Targets
IC50
HER2 HDAC EGFR
15.7 nM 4.4 nM 2.4 nM


Preparing Stock Solutions

Concentration Volume (DMSO) Mass 1 mg 5 mg 10 mg
1 mM 1.5686 mL 7.8430 mL 15.6860 mL
5 mM 0.3137 mL 1.5686 mL 3.1372 mL
10 mM 0.1569 mL 0.7843 mL 1.5686 mL
50 mM 0.0314 mL 0.1569 mL 0.3137 mL


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