Description：

GSK923295 is a first-in-class, specific allosteric inhibitor of CENP-E kinesin motor ATPase with K_i of 3.2 nM, and less potent to mutant I182 and T183. Phase 1.

Chemical Information：

Molecular Weight (MW)		592.13
Formula		C32H38ClN5O4
CAS No.		1088965-37-0
Solubility (25°C) *	DMSO	100 mg/mL (168.88 mM)
	Water	Insoluble
	Alcohol	100 mg/mL (168.88 mM)

Biological Activity：

Targets IC50

p38 MAPKα 4 - 20 nM

Preparing Stock Solutions

Concentration Volume (DMSO) Mass	1 mg	5 mg	10 mg
1 mM	1.6888 mL	8.4441 mL	16.8882 mL
5 mM	0.3378 mL	1.6888 mL	3.3776 mL
10 mM	0.1689 mL	0.8444 mL	1.6888 mL
50 mM	0.0338 mL	0.1689 mL	0.3378 mL

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