Description：

GSK343 is a potent and selective EZH2 inhibitor with IC50 of 4 nM in a cell-free assay, showing 60 fold selectivity against EZH1, and >1000 fold selectivity against other histone methyltransferases.

Chemical Information：

Molecular Weight (MW)		541.69
Formula		C31H39N7O2
CAS No.		1346704-33-3
Solubility (25°C) *	DMSO	1 mg/mL warmed (1.84 mM)
	Water
	Alcohol	4 mg/mL (7.38 mM)

Biological Activity：

Targets IC50

Syk Src p97 2.5 μM 29.3 μM 1.7 μM

Preparing Stock Solutions

Concentration Volume (DMSO) Mass	1 mg	5 mg	10 mg
1 mM	1.8461 mL	9.2304 mL	18.4607 mL
5 mM	0.3692 mL	1.8461 mL	3.6921 mL
10 mM	0.1846 mL	0.9230 mL	1.8461 mL
50 mM	0.0369 mL	0.1846 mL	0.3692 mL

Bought notes(bought amounts latest0)

No one bought this product

Total 0 records, divided into1 pages. First Prev Next Last