Description：

GSK J4 HCl is a cell permeable prodrug of GSK J1, which is the first selective inhibitor of the H3K27 histone demethylase JMJD3 and UTX with IC50 of 60 nM in a cell-free assay and inactive against a panel of demethylases of the JMJ family.

Chemical Information：

Molecular Weight (MW)		453.96
Formula		C24H27N5O2.HCl
CAS No.		1373423-53-0(free base)
Solubility (25°C) *	DMSO	90 mg/mL warmed (198.25 mM)
	Water	90 mg/mL (198.25 mM)
	Alcohol	90 mg/mL warmed (198.25 mM)

Preparing Stock Solutions

Concentration Volume (DMSO) Mass	1 mg	5 mg	10 mg
1 mM	2.2028 mL	11.0142 mL	22.0284 mL
5 mM	0.4406 mL	2.2028 mL	4.4057 mL
10 mM	0.2203 mL	1.1014 mL	2.2028 mL
50 mM	0.0441 mL	0.2203 mL	0.4406 mL

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