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Eltanexor (KPT-8602)

Eltanexor (KPT-8602)

Catalog Number: CC8553 Rank: comment rank 5

Size Price Qty
$ 102.00
$ 207.00
$ 553.00
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Description:

Eltanexor(KPT-8602) is a second-generation, orally bioavailable XPO1 inhibitor with IC50 values of 20−211 nM in 10 AML lines after 3 days exposure.

Chemical Information:

Molecular Weight (MW) 428.29
Formula

 

C17H10F6N6O

 

CAS No. 1642300-52-4
Solubility (25°C) * DMSO 85 mg/mL warmed (198.46 mM)
Water Insoluble
Alcohol 1 mg/mL warmed (2.33 mM)


Biological Activity:

Targets
IC50
WKY-E SHR-E
162.5 nM 170.3 nM


Preparing Stock Solutions

Concentration Volume (DMSO) Mass 1 mg 5 mg 10 mg
1 mM 2.3349 mL 11.6743 mL 23.3487 mL
5 mM 0.4670 mL 2.3349 mL 4.6697 mL
10 mM 0.2335 mL 1.1674 mL 2.3349 mL
50 mM 0.0467 mL 0.2335 mL 0.4670 mL


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