Search  
Your Position: Home > Protein Tyrosine Kinase > IGF-1R inhibitor > BMS-754807
All Categories
BMS-754807

BMS-754807

Catalog Number: CC1280 Rank: comment rank 5

Size Price Qty
$ 125.00
$ 189.00
$ 539.00
Total:
    
ChecmCatch Tel: 021-65878381 QQ Online
Email: kelvinyeng@hotmail.com    info@chemcatch.cn

Goods Info

Releate

Other

Description:

BMS-754807 is a potent and reversible inhibitor of IGF-1R/InsR with IC50 of 1.8 nM/1.7 nM in cell-free assays, less potent to Met, Aurora A/B, TrkA/B and Ron, and shows little activity to Flt3, Lck, MK2, PKA, PKC etc. Phase 2.

Chemical Information:

Molecular Weight (MW) 461.49
Formula

 

C23H24FN9O

 

CAS No. 1001350-96-4
Solubility (25°C) * DMSO 92 mg/mL (199.35 mM)
Water Insoluble
Alcohol 92 mg/mL (199.35 mM)


Biological Activity:

Targets
IC50
VEGFR2
1 nM


Preparing Stock Solutions

Concentration Volume (DMSO) Mass 1 mg 5 mg 10 mg
1 mM 2.1669 mL 10.8345 mL 21.6689 mL
5 mM 0.4334 mL 2.1669 mL 4.3338 mL
10 mM 0.2167 mL 1.0834 mL 2.1669 mL
50 mM 0.0433 mL 0.2167 mL 0.4334 mL


Bought notes(bought amounts latest0)

No one bought this product
Total 0 records, divided into1 pages. First Prev Next Last
Chem Catch products are for research use only. Not for human use. We do not sell to patients.

沪ICP备16042327号-2