Description：

BI2536 is a potent Plk1 inhibitor with IC50 of 0.83 nM in a cell-free assay. It shows 4- and 11-fold greater selectivity against Plk2 and Plk3. Phase 2.

Chemical Information：

Molecular Weight (MW)		521.66
Formula		C28H39N7O3
CAS No.		755038-02-9
Solubility (25°C) *	DMSO	21 mg/mL (40.25 mM)
	Water	Insoluble
	Alcohol	100 mg/mL (191.69 mM)

Biological Activity：

Targets IC50

ERα Erβ 23 nM 89 nM

Preparing Stock Solutions

Concentration Volume (DMSO) Mass	1 mg	5 mg	10 mg
1 mM	1.9170 mL	9.5848 mL	19.1696 mL
5 mM	0.3834 mL	1.9170 mL	3.8339 mL
10 mM	0.1917 mL	0.9585 mL	1.9170 mL
50 mM	0.0383 mL	0.1917 mL	0.3834 mL

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