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Selumetinib (AZD6244)

Selumetinib (AZD6244)

Catalog Number: CC1164 Rank: comment rank 5

Size Price Qty
$ 118.00
$ 259.00
$ 91.00
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Description:

Selumetinib (AZD6244) is a potent, highly selective MEK1 inhibitor with IC50 of 14 nM in cell-free assays, also inhibits ERK1/2 phosphorylation with IC50 of 10 nM, no inhibition to p38α, MKK6, EGFR, ErbB2, ERK2, B-Raf, etc. Phase 3.

Chemical Information:

Molecular Weight (MW) 457.68
Formula

 

C17H15BrClFN4O3

 

CAS No. 606143-52-6
Solubility (25°C) * DMSO 91 mg/mL warmed (198.82 mM)
Water Insoluble
Alcohol Insoluble


Preparing Stock Solutions

Concentration Volume (DMSO) Mass 1 mg 5 mg 10 mg
1 mM 2.1849 mL 10.9247 mL 21.8493 mL
5 mM 0.4370 mL 2.1849 mL 4.3699 mL
10 mM 0.2185 mL 1.0925 mL 2.1849 mL
50 mM 0.0437 mL 0.2185 mL 0.4370 mL


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