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Ki16198

Ki16198

Catalog Number: CC3062 Rank: comment rank 5

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Description:

Ki16198 is the methyl ester of Ki16425, which is a LPA antagonist and inhibits LPA1- and LPA3-induced inositol phosphate production with Ki of 0.34 μM and 0.93 μM, respectively, shows weaker inhibition for LPA2, no activity at LPA4, LPA5, LPA6.

Chemical Information:

Molecular Weight (MW) 488.98
Formula

 

C24H25ClN2O5S

 

CAS No. 355025-13-7
Solubility (25°C) * DMSO 96 mg/mL (196.32 mM)
Water Insoluble
Alcohol 35 mg/mL (71.57 mM)


Biological Activity:

Targets
IC50
PI3Kα PI3Kβ DNA-PK PI3Kδ
4 nM 0.5 nM 8.6 nM 0.1 nM


Preparing Stock Solutions

Concentration Volume (DMSO) Mass 1 mg 5 mg 10 mg
1 mM 2.0451 mL 10.2254 mL 20.4507 mL
5 mM 0.4090 mL 2.0451 mL 4.0901 mL
10 mM 0.2045 mL 1.0225 mL 2.0451 mL
50 mM 0.0409 mL 0.2045 mL 0.4090 mL


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