Description：

HER2-Inhibitor-1 is a potent and selective HER2 inhibitor with IC50 of 8 nM, equipotent against truncated p95-HER2, 500-fold more selective for HER2 versus EGFR. Phase 1.

Chemical Information：

Molecular Weight (MW)		569.63
Formula		C29H27N7O4S
CAS No.		937265-83-3
Solubility (25°C) *	DMSO	100 mg/mL (175.55 mM)
	Water	Insoluble
	Alcohol	3 mg/mL (5.26 mM)

Biological Activity：

Targets IC50

αvβ5 receptor αvβ3 receptor 79 nM 4.1 nM

Preparing Stock Solutions

Concentration Volume (DMSO) Mass	1 mg	5 mg	10 mg
1 mM	1.7555 mL	8.7776 mL	17.5553 mL
5 mM	0.3511 mL	1.7555 mL	3.5111 mL
10 mM	0.1756 mL	0.8778 mL	1.7555 mL
50 mM	0.0351 mL	0.1756 mL	0.3511 mL

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