Description：

GSK256066 is a selective PDE4B(equal affinity to isoforms A-D) inhibitor with IC50 of 3.2 pM, >380,000-fold selectivity versus PDE1/2/3/5/6 and >2500-fold selectivity against PDE4B versus PDE7.Phase 2.

Chemical Information：

Molecular Weight (MW)		518.58
Formula		C27H26N4O5S
CAS No.		801312-28-7
Solubility (25°C) *	DMSO	5 mg/mL (9.64 mM)
	Water	Insoluble
	Alcohol	Insoluble

Biological Activity：

Targets IC50

NF-κB 11 nM

Preparing Stock Solutions

Concentration Volume (DMSO) Mass	1 mg	5 mg	10 mg
1 mM	1.9283 mL	9.6417 mL	19.2834 mL
5 mM	0.3857 mL	1.9283 mL	3.8567 mL
10 mM	0.1928 mL	0.9642 mL	1.9283 mL
50 mM	0.0386 mL	0.1928 mL	0.3857 mL

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