Description：

GSK180736A, developed as a Rho-associated, coiled-coil-containing protein kinase inhibitor, binds to GRK2(G protein-coupled receptor kinase 2) with logIC50 pf -6.6 (logIC50 -4.0 for GRK5 and >-3 for GRK1); ≥400-fold selective for GRK2 over both GRK1 and GRK5.

Chemical Information：

Molecular Weight (MW)		365.36
Formula		C19H16FN5O2
CAS No.		817194-38-0
Solubility (25°C) *	DMSO	73 mg/mL warmed (199.8 mM)
	Water	Insoluble
	Alcohol	3 mg/mL warmed (8.21 mM)

Preparing Stock Solutions

Concentration Volume (DMSO) Mass	1 mg	5 mg	10 mg
1 mM	2.7370 mL	13.6851 mL	27.3703 mL
5 mM	0.5474 mL	2.7370 mL	5.4741 mL
10 mM	0.2737 mL	1.3685 mL	2.7370 mL
50 mM	0.0547 mL	0.2737 mL	0.5474 mL

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