Description：

Galeterone is a selective CYP17 inhibitor and androgen receptor (AR) antagonist with IC50 of 300 nM and 384 nM, respectively, and is a potent inhibitor of human prostate tumor growth. Phase 2.

Chemical Information：

Molecular Weight (MW)		388.55
Formula		C26H32N2O
CAS No.		851983-85-2
Solubility (25°C) *	DMSO	24 mg/mL (61.76 mM)
	Water	Insoluble
	Alcohol	40 mg/mL warmed (102.94 mM)

Biological Activity：

Targets IC50

5-HT(4b) 5-HT(4a) 8 nM 2.5 nM

Preparing Stock Solutions

Concentration Volume (DMSO) Mass	1 mg	5 mg	10 mg
1 mM	2.5737 mL	12.8684 mL	25.7367 mL
5 mM	0.5147 mL	2.5737 mL	5.1473 mL
10 mM	0.2574 mL	1.2868 mL	2.5737 mL
50 mM	0.0515 mL	0.2574 mL	0.5147 mL

Bought notes(bought amounts latest0)

No one bought this product

Total 0 records, divided into1 pages. First Prev Next Last