Description：

FR 180204 is an ATP-competitive, selective ERK inhibitor with Ki of 0.31 μM and 0.14 μM for ERK1 And ERK2, respectively. It is 30-fold less potent against the related kinase p38α and failed to inhibit any kinases(MEK1, MKK4, IKKα, PKCα, Src, Syc, and PDGFα) at less than 30 μM.

Chemical Information：

Molecular Weight (MW)		327.34
Formula		C18 H13 N7
CAS No.		865362-74-9
Solubility (25°C) *	DMSO	65 mg/mL (198.57 mM)
	Water	Insoluble
	Alcohol	2 mg/mL warmed (6.1 mM)

Preparing Stock Solutions

Concentration Volume (DMSO) Mass	1 mg	5 mg	10 mg
1 mM	3.0549 mL	15.2746 mL	30.5493 mL
5 mM	0.6110 mL	3.0549 mL	6.1099 mL
10 mM	0.3055 mL	1.5275 mL	3.0549 mL
50 mM	0.0611 mL	0.3055 mL	0.6110 mL

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